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1

Functionally biased modulation of A3 adenosine receptor agonist efficacy and potency by imidazoquinolinamine allosteric enhancers

Zhan-Guo Gao, Dennis Verzijl, Annelien Zweemer, Kai Ye, Anikó Göblyös, Adriaan P. IJzerman, Kenneth A. Jacobson

Journal:

Biochemical Pharmacology

Year:

2011

Language:

english

File:

PDF, 1.30 MB

english, 2011

2

A Series of 2,4-Disubstituted Quinolines as a New Class of Allosteric Enhancers of the Adenosine A 3 Receptor

Heitman, Laura H., Göblyös, Anikó, Zweemer, Annelien M., Bakker, Renée, Mulder-Krieger, Thea, van Veldhoven, Jacobus P. D., de Vries, Henk, Brussee, Johannes, IJzerman, Adriaan P.

Journal:

Journal of Medicinal Chemistry

Year:

2009

Language:

english

File:

PDF, 148 KB

english, 2009

3

Structure–Kinetic Relationships—An Overlooked Parameter in Hit-to-Lead Optimization: A Case of Cyclopentylamines as Chemokine Receptor 2 Antagonists

Vilums, Maris, Zweemer, Annelien J. M., Yu, Zhiyi, de Vries, Henk, Hillger, Julia M., Wapenaar, Hannah, Bollen, Ilse A. E., Barmare, Farhana, Gross, Raymond, Clemens, Jeremy, Krenitsky, Paul, Brussee,

Journal:

Journal of Medicinal Chemistry

Year:

2013

Language:

english

File:

PDF, 654 KB

english, 2013

4

Bias in chemokine receptor signalling

Zweemer, Annelien J.M., Toraskar, Jimita, Heitman, Laura H., IJzerman, Adriaan P.

Journal:

Trends in Immunology

Year:

2014

Language:

english

File:

PDF, 1.94 MB

english, 2014

5

False Positives in a Reporter Gene Assay: Identification and Synthesis of Substituted N -Pyridin-2-ylbenzamides as Competitive Inhibitors of Firefly Luciferase

Heitman, Laura H., van Veldhoven, Jacobus P. D., Zweemer, Annelien M., Ye, Kai, Brussee, Johannes, IJzerman, Adriaan P.

Journal:

Journal of Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 348 KB

english, 2008

6

Synthesis, binding affinity and structure–activity relationships of novel, selective and dual targeting CCR2 and CCR5 receptor antagonists

Junker, Anna, Kokornaczyk, Artur K., Zweemer, Annelien J. M., Frehland, Bastian, Schepmann, Dirk, Yamaguchi, Junichiro, Itami, Kenichiro, Faust, Andreas, Hermann, Sven, Wagner, Stefan, Schäfers, Micha

Journal:

Organic & Biomolecular Chemistry

Year:

2015

Language:

english

File:

PDF, 384 KB

english, 2015

7

When structure–affinity relationships meet structure–kinetics relationships: 3-((Inden-1-yl)amino)-1-isopropyl-cyclopentane-1-carboxamides as CCR2 antagonists

Vilums, Maris, Zweemer, Annelien J.M., Barmare, Farhana, van der Gracht, Anouk M.F., Bleeker, Dave C.T., Yu, Zhiyi, de Vries, Henk, Gross, Raymond, Clemens, Jeremy, Krenitsky, Paul, Brussee, Johannes,

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 1.29 MB

english, 2015

8

Synthesis and biological evaluation of spirocyclic antagonists of CCR2 (chemokine CC receptor subtype 2)

Strunz, Ann Kathrin, Zweemer, Annelien J.M., Weiss, Christina, Schepmann, Dirk, Junker, Anna, Heitman, Laura H., Koch, Michael, Wünsch, Bernhard

Journal:

Bioorganic & Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 890 KB

english, 2015

9

The AXL Receptor Is a Sensor of Ligand Spatial Heterogeneity

Meyer, Aaron S., Zweemer, Annelien J.M., Lauffenburger, Douglas A.

Journal:

Year:

2015

Language:

english

File:

PDF, 3.21 MB

english, 2015

10

Evaluation of (4-Arylpiperidin-1-yl)cyclopentanecarboxamides As High-Affinity and Long-Residence-Time Antagonists for the CCR2 Receptor

Vilums, Maris, Zweemer, Annelien J. M., Dilanchian, Arian, van Veldhoven, Jacobus P. D., de Vries, Henk, Brussee, Johannes, Saunders, John, Stamos, Dean, Heitman, Laura H., IJzerman, Adriaan P.

Journal:

Year:

2015

Language:

english

File:

PDF, 518 KB

english, 2015

11

Apoptotic Bodies Elicit Gas6-mediated Migration of AXL-expressing Tumor Cells

Zweemer, Annelien JM, French, Cory B, Mesfin, Joshua, Gordonov, Simon, Meyer, Aaron S, Lauffenburger, Douglas A.

Journal:

Molecular Cancer Research

Year:

2017

Language:

english

File:

PDF, 7.97 MB

english, 2017

12

A two-state model for the kinetics of competitive radioligand binding

Guo, Dong, Peletier, Lambertus A, Bridge, Lloyd, Keur, Wesley, de Vries, Henk, Zweemer, Annelien, Heitman, Laura H, IJzerman, Adriaan P

Journal:

British Journal of Pharmacology

Year:

2018

Language:

english

File:

PDF, 1.44 MB

english, 2018

13

Pyrrolone derivatives as intracellular allosteric modulators for chemokine receptors: Selective and dual-targeting inhibitors of CC Chemokine Receptors 1 and 2

Ortiz Zacarías, Natalia Veneranda, van Veldhoven, Jacobus P. D., Portner, Laura, van Spronsen, Eric, Ullo, Salviana, Veenhuizen, Margo, van der Velden, Wijnand J.C., Zweemer, Annelien J.M., Kreekel, R

Journal:

Journal of Medicinal Chemistry

Year:

2018

Language:

english

File:

PDF, 1.96 MB

english, 2018

14

Metastasis: crosstalk between tissue mechanics and tumour cell plasticity

Coban, Bircan, Bergonzini, Cecilia, Zweemer, Annelien J. M., Danen, Erik H. J.

Journal:

British Journal of Cancer

Year:

2020

File:

PDF, 1.24 MB

2020

15

Development of the First Potential Nonpeptidic Positron Emission Tomography Tracer for the Imaging of CCR2 Receptors

Wagner, Stefan, Moura Gatti, Fernando, Silva, Daniel G., Ortiz Zacarias, Natalia V., Zweemer, Annelien J. M., Hermann, Sven, De Maria, Monica, Koch, Michael, Weiss, Christina, Schepmann, Dirk, Heitman

Journal:

Year:

2020

File:

PDF, 1.24 MB

2020